Selected article for: "antimalarial agent and vitro activity"

Author: Ishiyama, Aki; Hokari, Rei; Nonaka, Kenichi; Chiba, Takuya; Miura, Hiromi; Otoguro, Kazuhiko; Iwatsuki, Masato
Title: Diatretol, an α, α′-dioxo-diketopiperazine, is a potent in vitro and in vivo antimalarial
  • Cord-id: fsmiw3o4
  • Document date: 2021_1_14
  • ID: fsmiw3o4
    Snippet: A fungal metabolite, diatretol, has shown to be a promising antimalarial agent. Diatretol displayed potent in vitro antiparasitic activity against the Plasmodium falciparum K1 strain, with an IC(50) value of 378 ng ml(−1), as well as in vivo efficacy in a Plasmodium berghei-infected mice model, with ca. 50% inhibition at 30 mg/kg (p.o.).
    Document: A fungal metabolite, diatretol, has shown to be a promising antimalarial agent. Diatretol displayed potent in vitro antiparasitic activity against the Plasmodium falciparum K1 strain, with an IC(50) value of 378 ng ml(−1), as well as in vivo efficacy in a Plasmodium berghei-infected mice model, with ca. 50% inhibition at 30 mg/kg (p.o.).

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